SCHEMBL7006426

SCHEMBL7006426

O=C(NC(CC1CCCCC1)C(=O)N([C@H]1CCCNCC1=O)S(=O)(=O)c1ccccn1)c1ccco1

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSK P43235 15/20 0.53
CTSL P07711 14/20 0.53
CTSS P25774 14/20 0.53
ALDH1A1 P00352 2/20 0.39
USP30 Q70CQ3 1/20 0.37
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6214223 0.88 CTSK (0.56) CTSKCTSLCTSSALDH1A1USP30
SCHEMBL7009811 0.88 CTSK (0.46) CTSKCTSLCTSS
SCHEMBL7011830 0.88 CTSL (0.40) CTSKCTSLCTSSUSP30
SCHEMBL7006137 0.87 CTSL (0.39) CTSKCTSLCTSSUSP30
SCHEMBL6073049 0.87 CTSK (0.39) CTSKCTSLCTSSUSP30
SCHEMBL6073055 0.86 CTSL (0.42) CTSKCTSLCTSSUSP30
SCHEMBL7012868 0.86 CTSS (0.40) CTSKCTSLCTSSUSP30
SCHEMBL6072667 0.85 CTSK (0.41) CTSKCTSLCTSSUSP30
SCHEMBL7011520 0.85 CTSS (0.39) CTSKCTSLCTSSUSP30
SCHEMBL6072616 0.85 CTSK (0.40) CTSKCTSLCTSSUSP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1278502-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-05-21 EP claimed
EP-1278502-A2 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-01-29 EP claimed
WO-2001089451-A2 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-11-29 WO claimed
EP-1278502-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-05-21 EP disclosed
EP-1278502-A2 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-01-29 EP disclosed
WO-2001089451-A2 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-11-29 WO disclosed