SCHEMBL7008944

SCHEMBL7008944

Cc1cccc2nc(CCc3ccc(C(=O)c4ccc(O)cc4)cc3)n(C)c(=O)c12

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CASR P41180 2/20 0.45
GFER P55789 1/20 0.42
PIK3CD O00329 2/20 0.42
HDAC6 Q9UBN7 2/20 0.40
NTRK1 P04629 7/20 0.39
NTRK2 Q16620 6/20 0.39
NPC1 O15118 1/20 0.39
GAA P10253 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HDAC8 Q9BY41 1/20 0.38
TRPA1 O75762 1/20 0.38
PARP1 P09874 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7012231 0.90 TRPA1 (0.48) CASRPIK3CDHDAC6NTRK1NTRK2
SCHEMBL7015330 0.88 NTRK1 (0.46) CASRPIK3CDHDAC6NTRK1NTRK2
Hydrochloric Acid SCHEMBL7014173 0.82 HRH3 (0.40) CASRGAASMN1; SMN2
SCHEMBL7015787 0.81 MEN1 (0.51) CASRHDAC6NPC1SMN1; SMN2HDAC8
Hydrochloric Acid SCHEMBL7017276 0.79 LSS (0.35) CASRPIK3CDHDAC6NTRK1NTRK2
Hydrochloric Acid SCHEMBL7018696 0.79 KMT2A (0.43) CASRPIK3CDHDAC6NPC1GAA
SCHEMBL7011506 0.76 MEN1 (0.55) HDAC6SMN1; SMN2HDAC8
SCHEMBL7019291 0.75 CASR (0.43) CASRRAB9ASMN1; SMN2
SCHEMBL7019084 0.74 MAOA (0.46) CASRSMN1; SMN2TRPA1
SCHEMBL7013546 0.74 MAOA (0.47) PIK3CDHDAC6NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed