SCHEMBL7013546

SCHEMBL7013546

Cc1cccc2nc(CSc3ccc(C(=O)c4ccc(Cl)cc4)cc3)n(C)c(=O)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.47
MAOB P27338 3/20 0.47
KMT2A Q03164 4/20 0.43
NPSR1 Q6W5P4 3/20 0.43
MAPT P10636 3/20 0.43
MEN1 O00255 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
HDAC6 Q9UBN7 1/20 0.41
LMNA P02545 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
TSHR P16473 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
USP2 O75604 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PIK3CG P48736 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7012231 0.83 TRPA1 (0.48) NPSR1MAPTCYP1A2CYP2D6CYP2C9
SCHEMBL7018370 0.82 MEN1 (0.50) MAOAMAOBKMT2ANPSR1MAPT
SCHEMBL7018222 0.79 TDP1 (0.49) MAOAMAOBKMT2ANPSR1MAPT
SCHEMBL7019084 0.76 MAOA (0.46) MAOAMAOBKMT2ANPSR1MAPT
SCHEMBL7011506 0.75 MEN1 (0.55) KMT2AMAPTMEN1CYP1A2CYP2D6
SCHEMBL7014766 0.75 NPC1 (0.58) MAOBKMT2ANPSR1MAPTCYP1A2
SCHEMBL7014764 0.75 NPC1 (0.58) MAOBKMT2ANPSR1MAPTCYP1A2
SCHEMBL7014540 0.74 DRD2 (0.52) KMT2ANPSR1MAPTMEN1CYP1A2
SCHEMBL7008944 0.74 CASR (0.45) HDAC6SMN1; SMN2TRPA1PIK3CDNPC1
SCHEMBL7101327 0.73 MEN1 (0.60) KMT2AMAPTMEN1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed