SCHEMBL7009003

SCHEMBL7009003

Clc1ccc(CC(Br)c2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.47
CHRNB2 P17787 1/20 0.45
CHRNA4 P43681 1/20 0.45
SLC6A2 P23975 2/20 0.44
SLC6A3 Q01959 2/20 0.44
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
IDO1 P14902 2/20 0.41
TDO2 P48775 2/20 0.41
SIGMAR1 Q99720 1/20 0.41
CNR1 P21554 6/20 0.41
CNR2 P34972 6/20 0.41
PPARG P37231 2/20 0.40
PPARA Q07869 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1641620 0.85 SLC6A2 (0.48) SLC6A4SLC6A2SLC6A3CYP1A2CYP2D6
SCHEMBL7005600 0.79 PNMT (0.53) SLC6A4SLC6A2IDO1TDO2SIGMAR1
SCHEMBL25343509 0.78 SMO (0.53) SLC6A4CHRNB2CHRNA4SLC6A2SLC6A3
SCHEMBL16745473 0.78 FFAR1 (0.45) SLC6A4SLC6A2SLC6A3SIGMAR1PPARG
SCHEMBL6442526 0.76 SLC6A4 (0.57) SLC6A4CHRNB2CHRNA4SLC6A2SLC6A3
SCHEMBL4603704 0.76 SLC6A2 (0.53) SLC6A4CHRNB2CHRNA4SLC6A2SLC6A3
SCHEMBL4603712 0.76 SLC6A2 (0.53) SLC6A4CHRNB2CHRNA4SLC6A2SLC6A3
SCHEMBL8317452 0.76 ALDH1A1 (0.45) SLC6A4SLC6A2SLC6A3CNR1CNR2
Ammonia Solution, Strong SCHEMBL8867131 0.74 SLC6A2 (0.52) SLC6A4CHRNB2CHRNA4SLC6A2SLC6A3
SCHEMBL3374924 0.74 SLC6A2 (0.56) SLC6A4CHRNB2CHRNA4SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1267906-A1 LACTAMS AS INHIBITORS OF A-BETA PROTEIN PRODUCTION Bristol-Myers Squibb Pharma Company (US) 2003-01-02 EP claimed
WO-2001072324-A1 LACTAMS AS INHIBITORS OF A-BETA PROTEIN PRODUCTION BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2001-10-04 WO claimed