SCHEMBL8317452

SCHEMBL8317452

FC(F)(F)c1ccc(CC(Br)c2ccccc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
PDPK1 O15530 1/20 0.44
PPARG P37231 1/20 0.44
PPARA Q07869 1/20 0.44
KIF11 P52732 1/20 0.44
ACP3 P15309 3/20 0.44
SLC6A9 P48067 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SLC6A2 P23975 2/20 0.42
SLC6A4 P31645 2/20 0.42
SLC6A3 Q01959 2/20 0.42
KCNK2 O95069 1/20 0.42
KCNH2 Q12809 1/20 0.42
CACNA1C Q13936 1/20 0.42
CNR2 P34972 1/20 0.41
FPR2 P25090 1/20 0.40
PTPN1 P18031 1/20 0.40
CNR1 P21554 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2312292 0.82 PDPK1 (0.48) ALDH1A1TSHRPDPK1PPARGPPARA
SCHEMBL1641620 0.80 SLC6A2 (0.48) ALDH1A1TSHRACP3SLC6A2SLC6A4
SCHEMBL8875932 0.79 ALDH1A1 (0.45) ALDH1A1TSHRPDPK1PPARGPPARA
SCHEMBL3128823 0.77 TAAR1 (0.48) ALDH1A1PPARGPPARAKIF11PTPN1
SCHEMBL9733971 0.76 SLC6A9 (0.50) ALDH1A1TSHRPPARGPPARAKIF11
SCHEMBL7009003 0.76 SLC6A4 (0.47) PPARGPPARASLC6A2SLC6A4SLC6A3
SCHEMBL7523008 0.75 ACP3 (0.55) ALDH1A1TSHRPDPK1KIF11ACP3
SCHEMBL21085616 0.75 BACE1 (0.47) ALDH1A1TSHRPPARGPPARAKIF11
SCHEMBL28604259 0.75 ESR2 (0.51) ALDH1A1TSHRPDPK1PPARGPPARA
SCHEMBL5755207 0.73 PPARG (0.43) PPARGPPARAACP3SLC6A9SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929534-A1 TRYCYCLIC COMPOUNDS AS PROSTAGLANDIN I2 RECEPTOR AGONISTS Takeda Pharmaceutical Company Limited (JP) 1999-07-21 EP disclosed
WO-1998013356-A1 TRYCYCLIC COMPOUNDS AS PROSTAGLANDIN I2 RECEPTOR AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-04-02 WO disclosed