SCHEMBL7009560

SCHEMBL7009560

CCOC(=O)/C(=C\Nc1c(F)cc(F)cc1F)C(=O)c1cc(F)c(Cl)nc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 5/20 0.41
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
MEN1 O00255 5/20 0.40
KMT2A Q03164 5/20 0.40
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
NPY1R P25929 1/20 0.39
NPY2R P49146 1/20 0.39
MAPT P10636 5/20 0.38
DHODH Q02127 4/20 0.38
GAA P10253 3/20 0.38
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
MAPK1 P28482 1/20 0.37
LMNA P02545 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7009563 1.00 NPSR1 (0.41) NPSR1KEAP1NFE2L2MEN1KMT2A
SCHEMBL5258270 0.86 MEN1 (0.43) NPSR1KEAP1NFE2L2MEN1KMT2A
SCHEMBL5258272 0.86 MEN1 (0.43) NPSR1KEAP1NFE2L2MEN1KMT2A
SCHEMBL9537592 0.86 DHODH (0.51) NPSR1MEN1KMT2AKDM4EALDH1A1
SCHEMBL14700370 0.85 KEAP1 (0.44) NPSR1KEAP1NFE2L2MEN1KMT2A
SCHEMBL9536539 0.84 DHODH (0.53) NPSR1KEAP1NFE2L2MEN1KMT2A
SCHEMBL9535935 0.83 DHODH (0.50) NPSR1MEN1KMT2AKDM4EALDH1A1
SCHEMBL8129004 0.83 NPSR1 (0.57) NPSR1KEAP1NFE2L2MEN1KMT2A
SCHEMBL9684796 0.82 KEAP1 (0.42) NPSR1KEAP1NFE2L2MEN1KMT2A
SCHEMBL22774063 0.82 KEAP1 (0.42) NPSR1KEAP1NFE2L2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0787720-B1 PYRIDONECARBOXYLATE DERIVATIVE OR SALT THEREOF AND ANTIBACTERIAL CONTAINING THE SAME AS ACTIVE INGREDIENT WAKUNAGA SEIYAKU KK (JP) 2003-07-16 EP disclosed
US-5910498-A NOVEL COMPOUNDS HAVING REDUCED CYTOTOXICITY, PHOTOTOXICITY; TREATING BACTERIAL AND VIRAL INFECTIONS WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1999-06-08 US disclosed
EP-0787720-A1 NOVEL PYRIDONECARBOXYLATE DERIVATIVE OR SALT THEREOF AND ANTIBACTERIAL CONTAINING THE SAME AS ACTIVE INGREDIENT WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1997-08-06 EP disclosed