SCHEMBL7010932

SCHEMBL7010932

CCc1c(C)nc2n(Cc3ccc(C(=O)c4ccc(O)cc4)cc3)ccn2c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.42
TP53 P04637 3/20 0.39
MAPT P10636 3/20 0.39
HDAC6 Q9UBN7 3/20 0.38
HDAC3 O15379 2/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC2 Q92769 2/20 0.38
HDAC8 Q9BY41 1/20 0.38
TDP1 Q9NUW8 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
THRB P10828 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
POLB P06746 1/20 0.34
ENPP2 Q13822 1/20 0.34
CASR P41180 1/20 0.34
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
PIK3CD O00329 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016720 0.91 SRD5A2 (0.42) TP53MAPTHDAC6HDAC3HDAC1
SCHEMBL7015350 0.91 TP53 (0.44) TP53MAPTHDAC6HDAC3HDAC1
SCHEMBL7016860 0.87 KDM4E (0.43) MAPTHDAC6HDAC3HDAC1HDAC2
SCHEMBL7011674 0.86 RAB9A (0.39) TP53MAPTHDAC6HDAC3HDAC1
Hydrochloric Acid SCHEMBL7018460 0.84 CYP19A1 (0.41) CYP19A1MAPTKMT2AHTTSMN1; SMN2
SCHEMBL7016868 0.83 ENPP2 (0.42) TP53MAPTHDAC6HDAC3HDAC1
SCHEMBL7015591 0.81 MEN1 (0.50) TP53MAPTTHRBMEN1KMT2A
SCHEMBL7016621 0.80 TP53 (0.42) TP53MAPTHDAC6HDAC3HDAC1
SCHEMBL7014882 0.79 KDM4E (0.42) MAPTHDAC1HTTSMN1; SMN2
Hydrochloric Acid SCHEMBL7021475 0.79 L3MBTL3 (0.50) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed