SCHEMBL7012279

SCHEMBL7012279

Cn1c(SCc2ccc(C(=O)c3ccc(OCCN4CCCCC4)cc3)cc2)nc2ccsc2c1=O

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
PKM P14618 1/20 0.56
HTT P42858 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
PSMB1 P20618 1/20 0.53
PSMB5 P28074 1/20 0.53
PSMB2 P49721 1/20 0.53
LTA4H P09960 4/20 0.48
ESR1 P03372 2/20 0.44
ESR2 Q92731 2/20 0.44
BCHE P06276 4/20 0.44
ACHE P22303 4/20 0.44
LMNA P02545 2/20 0.43
KDM4E B2RXH2 3/20 0.43
GPR35 Q9HC97 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
MCHR1 Q99705 1/20 0.42
GCGR P47871 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7020967 0.92 ALDH1A1 (0.54) ALDH1A1PKMHTTSMN1; SMN2PSMB1
SCHEMBL7013586 0.83 SMN1; SMN2 (0.65) ALDH1A1PKMHTTSMN1; SMN2LMNA
Hydrochloric Acid SCHEMBL7020207 0.83 KCNH2 (0.50) ALDH1A1PSMB1PSMB5PSMB2LTA4H
SCHEMBL9051500 0.83 PSMB1 (0.50) ALDH1A1PSMB1PSMB5PSMB2LTA4H
Hydrochloric Acid SCHEMBL7018187 0.82 PSMB1 (0.49) PSMB1PSMB5PSMB2LTA4HESR1
Hydrochloric Acid SCHEMBL7012383 0.82 KCNH2 (0.51) ALDH1A1PSMB1PSMB5PSMB2LTA4H
SCHEMBL7015837 0.81 SMN1; SMN2 (0.70) ALDH1A1PKMHTTSMN1; SMN2LMNA
SCHEMBL7016121 0.80 SMN1; SMN2 (0.69) ALDH1A1PKMHTTSMN1; SMN2LMNA
SCHEMBL9052713 0.80 SMN1; SMN2 (0.69) ALDH1A1PKMHTTSMN1; SMN2LMNA
Hydrochloric Acid SCHEMBL7017180 0.79 KCNH2 (0.44) ALDH1A1PKMHTTSMN1; SMN2PSMB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed