SCHEMBL7012599

SCHEMBL7012599

CC(C)(C)[Si](C)(C)Oc1ccc(C(=O)c2ccc(CBr)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PREP P48147 4/20 0.43
ELANE P08246 5/20 0.42
SRD5A2 P31213 2/20 0.42
PPARG P37231 2/20 0.40
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
KMT2A Q03164 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
VNN1 O95497 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CA12 O43570 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2500559 0.89 ELANE (0.52) PREPELANEPPARGKMT2ANPSR1
SCHEMBL1601708 0.87 PREP (0.46) PREPELANEPPARGALDH1A1CA12
SCHEMBL20364920 0.83 LMNA (0.53) PREPELANESRD5A2KMT2ANPSR1
SCHEMBL5280416 0.83 ELANE (0.57) PREPELANESRD5A2PPARGALDH1A1
SCHEMBL5032713 0.80 GSK3B (0.59) PREPLMNAMAPK1ALDH1A1CA12
SCHEMBL3550962 0.78 MEN1 (0.49) PREPELANEKMT2ANPSR1MEN1
SCHEMBL2506528 0.78 SRD5A2 (0.46) PREPSRD5A2LMNAALDH1A1HTT
SCHEMBL5591858 0.77 RAB9A (0.65) CES2CES1KMT2ANPSR1MEN1
SCHEMBL936407 0.77 MAPT (0.53) PREPKMT2ANPSR1LMNAMAPT
SCHEMBL6542930 0.77 CA1 (0.52) PREPSRD5A2KMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed