SCHEMBL7014792

SCHEMBL7014792

COc1ccc(Cc2nc3ccccc3c(=O)n2-c2ccc(C(O)(C(F)(F)F)C(F)(F)F)cc2)cc1

nearest known ligand 0.74

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.74
MEN1 O00255 1/20 0.59
CYP1A2 P05177 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2D6 P10635 1/20 0.59
CYP2C9 P11712 1/20 0.59
CYP2C19 P33261 1/20 0.59
KMT2A Q03164 1/20 0.59
RAB9A P51151 2/20 0.56
NPC1 O15118 1/20 0.56
PDE10A Q9Y233 9/20 0.55
GAA P10253 1/20 0.54
LMNA P02545 1/20 0.50
NPSR1 Q6W5P4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7013129 0.91 ALDH1A1 (0.65) ALDH1A1MEN1CYP1A2CYP3A4CYP2D6
SCHEMBL7023261 0.90 ALDH1A1 (0.70) ALDH1A1MEN1CYP1A2CYP3A4CYP2D6
SCHEMBL7016256 0.90 ALDH1A1 (0.64) ALDH1A1MEN1CYP1A2CYP3A4CYP2D6
SCHEMBL7020221 0.90 ALDH1A1 (0.63) ALDH1A1MEN1CYP1A2CYP3A4CYP2D6
SCHEMBL7020429 0.89 ALDH1A1 (0.60) ALDH1A1MEN1CYP1A2CYP3A4CYP2D6
SCHEMBL7022684 0.89 ALDH1A1 (0.73) ALDH1A1MEN1KMT2ARAB9ANPC1
SCHEMBL7011889 0.89 ALDH1A1 (0.63) ALDH1A1KMT2ARAB9ANPC1LMNA
SCHEMBL7103501 0.88 ALDH1A1 (0.61) ALDH1A1MEN1KMT2ARAB9ANPC1
SCHEMBL7017881 0.88 ALDH1A1 (0.61) ALDH1A1MEN1KMT2ARAB9ANPC1
SCHEMBL7026336 0.87 ALDH1A1 (0.60) ALDH1A1KMT2ARAB9ANPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003106435-A1 FUSED-RING PYRIMIDIN-4(3H)-ONE DERIVATIVES, PROCESSES FOR THE PREPARATION AND USES THEREOF SANKYO COMPANY, LIMITED (JP) 2003-12-24 WO claimed
WO-2003106435-A1 FUSED-RING PYRIMIDIN-4(3H)-ONE DERIVATIVES, PROCESSES FOR THE PREPARATION AND USES THEREOF SANKYO COMPANY, LIMITED (JP) 2003-12-24 WO disclosed