SCHEMBL7013129

SCHEMBL7013129

COc1ccc2c(=O)n(-c3ccc(C(O)(C(F)(F)F)C(F)(F)F)cc3)c(Cc3ccccc3)nc2c1

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.65
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
PDE10A Q9Y233 7/20 0.51
CYP3A4 P08684 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
MEN1 O00255 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
KMT2A Q03164 1/20 0.49
NPSR1 Q6W5P4 1/20 0.46
USP2 O75604 1/20 0.46
HTR7 P34969 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7020221 0.94 ALDH1A1 (0.63) ALDH1A1NPC1RAB9APDE10ACYP3A4
SCHEMBL7014792 0.91 ALDH1A1 (0.74) ALDH1A1NPC1RAB9APDE10ACYP3A4
SCHEMBL7016256 0.90 ALDH1A1 (0.64) ALDH1A1NPC1RAB9APDE10ACYP3A4
SCHEMBL5062276 0.88 ALDH1A1 (0.55) ALDH1A1NPC1RAB9APDE10ANPSR1
SCHEMBL7025946 0.88 ALDH1A1 (0.57) ALDH1A1NPC1RAB9AKMT2ANPSR1
SCHEMBL7017650 0.88 ALDH1A1 (0.64) ALDH1A1NPC1RAB9APDE10AKMT2A
SCHEMBL7019930 0.86 ALDH1A1 (0.56) ALDH1A1NPC1RAB9ACYP3A4CYP2C9
SCHEMBL7017695 0.86 ALDH1A1 (0.53) ALDH1A1NPC1RAB9APDE10ACYP3A4
SCHEMBL7015149 0.86 ALDH1A1 (0.53) ALDH1A1NPC1RAB9APDE10ACYP3A4
SCHEMBL7023261 0.86 ALDH1A1 (0.70) ALDH1A1NPC1RAB9APDE10ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003106435-A1 FUSED-RING PYRIMIDIN-4(3H)-ONE DERIVATIVES, PROCESSES FOR THE PREPARATION AND USES THEREOF SANKYO COMPANY, LIMITED (JP) 2003-12-24 WO claimed
WO-2003106435-A1 FUSED-RING PYRIMIDIN-4(3H)-ONE DERIVATIVES, PROCESSES FOR THE PREPARATION AND USES THEREOF SANKYO COMPANY, LIMITED (JP) 2003-12-24 WO disclosed