SCHEMBL7015308

SCHEMBL7015308

CC(CCNC(=O)c1ccc(OC(F)F)cc1)CC(=O)N1CCC2OCC(=O)C21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.46
CTSS P25774 4/20 0.42
CTSV O60911 3/20 0.41
CTSL P07711 3/20 0.41
KMT2A Q03164 1/20 0.40
ATM Q13315 2/20 0.39
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.35
IDO1 P14902 1/20 0.35
ALOX15 P16050 1/20 0.35
GFER P55789 1/20 0.35
ADAM17 P78536 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016550 0.95 CTSK (0.41) CTSKCTSSCTSVCTSLKMT2A
SCHEMBL4459438 0.91 CTSK (0.48) CTSKCTSSCTSVCTSLALDH1A1
SCHEMBL4451932 0.89 CTSK (0.47) CTSKCTSSCTSVCTSL
SCHEMBL4457938 0.88 CTSS (0.47) CTSKCTSSCTSVCTSLALDH1A1
SCHEMBL4452707 0.88 CTSK (0.50) CTSKCTSSCTSVCTSLKMT2A
SCHEMBL7018355 0.87 CTSK (0.52) CTSKCTSSCTSVCTSL
SCHEMBL4452660 0.87 CTSK (0.49) CTSKCTSSCTSVCTSLALDH1A1
SCHEMBL4452610 0.87 CTSK (0.49) CTSKCTSSCTSVCTSLNPC1
SCHEMBL4451610 0.87 CTSS (0.55) CTSKCTSSCTSVCTSLNPC1
SCHEMBL4452668 0.86 CTSK (0.62) CTSKCTSSCTSVCTSLALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362052-A1 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES Amura Therapeutics Limited (GB) 2003-11-19 EP disclosed
WO-2002057270-A1 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES AMURA THERAPEUTICS LIMITED (GB) 2002-07-25 WO disclosed