SCHEMBL7015451

SCHEMBL7015451

Cc1nc2n(Cc3ccc(C(=O)c4ccc(Cl)cc4Cl)cc3)ccn2c(=O)c1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.44
MAPT P10636 6/20 0.42
RAB9A P51151 1/20 0.42
TP53 P04637 3/20 0.41
TDP1 Q9NUW8 1/20 0.41
PIK3CD O00329 3/20 0.39
PIK3CB P42338 3/20 0.39
CHEK2 O96017 1/20 0.38
HDAC3 O15379 2/20 0.37
HDAC1 Q13547 2/20 0.37
HDAC2 Q92769 2/20 0.37
HDAC8 Q9BY41 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
POLB P06746 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CYP2C9 P11712 1/20 0.37
HTT P42858 2/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7015959 0.90 TP53 (0.44) MAPTRAB9ATP53TDP1PIK3CD
SCHEMBL7015342 0.83 MAPT (0.46) MAPTTP53TDP1PIK3CDPIK3CB
Hydrochloric Acid SCHEMBL7013530 0.80 L3MBTL1 (0.39) MAPTRAB9ATP53TDP1PIK3CD
SCHEMBL7015350 0.78 TP53 (0.44) MAPTRAB9ATP53TDP1PIK3CD
SCHEMBL7014282 0.77 TP53 (0.41) MAPTRAB9ATP53TDP1PIK3CD
SCHEMBL7016868 0.76 ENPP2 (0.42) MAPTRAB9ATP53TDP1PIK3CD
SCHEMBL7016044 0.74 PIK3CD (0.55) MAPTRAB9ATP53TDP1PIK3CD
SCHEMBL7016621 0.72 TP53 (0.42) MAPTTP53TDP1PIK3CDPIK3CB
SCHEMBL7016720 0.72 SRD5A2 (0.42) SRD5A2MAPTTP53TDP1HDAC3
SCHEMBL7010932 0.72 CYP19A1 (0.42) MAPTTP53TDP1PIK3CDPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed