SCHEMBL7015626

SCHEMBL7015626

Cn1c(=O)c2c(nc(Cl)n2Cc2ccc(C(=O)c3ccc(Cl)cc3)cc2)n(C)c1=O

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.67
SMN1; SMN2 Q16637 2/20 0.66
CYP1A2 P05177 2/20 0.66
CYP2C19 P33261 2/20 0.66
CYP3A4 P08684 1/20 0.66
CYP2C9 P11712 1/20 0.66
TSHR P16473 2/20 0.60
RAB9A P51151 1/20 0.60
MAPT P10636 5/20 0.59
ALDH1A1 P00352 4/20 0.59
NPSR1 Q6W5P4 4/20 0.59
MAPK1 P28482 2/20 0.59
ATM Q13315 1/20 0.57
TP53 P04637 2/20 0.54
MAOA P21397 1/20 0.53
MAOB P27338 1/20 0.53
LMNA P02545 2/20 0.53
RECQL P46063 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16029209 0.92 HTT (0.78) HTTSMN1; SMN2CYP1A2CYP2C19CYP3A4
SCHEMBL7017271 0.90 TSHR (0.59) HTTSMN1; SMN2CYP1A2CYP2C19CYP3A4
SCHEMBL7016485 0.88 ALDH1A1 (0.60) HTTSMN1; SMN2CYP1A2CYP2C19CYP3A4
SCHEMBL7016235 0.87 SMN1; SMN2 (0.63) HTTSMN1; SMN2TSHRRAB9AMAPT
SCHEMBL555962 0.82 HTT (0.74) HTTSMN1; SMN2CYP1A2CYP2C19CYP3A4
SCHEMBL555173 0.81 HTT (0.78) HTTSMN1; SMN2CYP1A2CYP2C19CYP3A4
SCHEMBL7015623 0.80 TSHR (0.56) HTTSMN1; SMN2TSHRRAB9AMAPT
SCHEMBL7017096 0.80 MAPK1 (0.53) HTTSMN1; SMN2TSHRRAB9AMAPT
SCHEMBL13083068 0.80 HTT (0.71) HTTSMN1; SMN2CYP1A2CYP2C19CYP3A4
SCHEMBL16028263 0.80 HPGD (0.62) HTTSMN1; SMN2CYP1A2CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed