SCHEMBL7017271

SCHEMBL7017271

Cc1nc2c(c(=O)n(C)c(=O)n2C)n1Cc1ccc(C(=O)c2ccc(Cl)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.59
RAB9A P51151 1/20 0.59
MAPT P10636 5/20 0.59
ALDH1A1 P00352 5/20 0.58
NPSR1 Q6W5P4 4/20 0.58
MAPK1 P28482 1/20 0.58
ATM Q13315 1/20 0.56
HTT P42858 3/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
LMNA P02545 1/20 0.54
TP53 P04637 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
PLD3 Q8IV08 1/20 0.53
MAOA P21397 1/20 0.52
MAOB P27338 1/20 0.52
POLB P06746 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7015623 0.90 TSHR (0.56) TSHRRAB9AMAPTALDH1A1NPSR1
SCHEMBL7015626 0.90 HTT (0.67) TSHRRAB9AMAPTALDH1A1NPSR1
SCHEMBL7016485 0.87 ALDH1A1 (0.60) TSHRRAB9AMAPTALDH1A1NPSR1
SCHEMBL7016235 0.86 SMN1; SMN2 (0.63) TSHRRAB9AMAPTALDH1A1NPSR1
SCHEMBL16664758 0.83 ALDH1A1 (0.67) TSHRRAB9AMAPTALDH1A1NPSR1
SCHEMBL16364219 0.82 TSHR (0.62) TSHRRAB9AMAPTALDH1A1NPSR1
SCHEMBL8646797 0.82 TSHR (0.49) TSHRRAB9AMAPTALDH1A1NPSR1
SCHEMBL18834914 0.81 TP53 (0.58) TSHRRAB9AMAPTALDH1A1NPSR1
SCHEMBL29256877 0.81 THRB (0.61) TSHRRAB9AMAPTALDH1A1NPSR1
SCHEMBL16029209 0.80 HTT (0.78) TSHRRAB9AMAPTALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed