SCHEMBL7016306

SCHEMBL7016306

CCn1c(SC)nc2c(ccn2Cc2ccc(C(=O)c3ccc(OC(C)N(C)C)cc3)cc2)c1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.35
MAPT P10636 1/20 0.35
P2RX3 P56373 2/20 0.35
HDAC1 Q13547 4/20 0.34
HDAC6 Q9UBN7 3/20 0.34
HDAC2 Q92769 3/20 0.34
HDAC3 O15379 2/20 0.34
HDAC4 P56524 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
RXFP1 Q9HBX9 3/20 0.33
TSHR P16473 2/20 0.33
ATM Q13315 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ALDH1A1 P00352 3/20 0.33
THRB P10828 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HPGD P15428 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016308 0.84 CYP19A1 (0.39) TP53MAPTP2RX3RXFP1TSHR
Hydrochloric Acid SCHEMBL7012709 0.84 SRC (0.37) TP53MAPTP2RX3HDAC1HDAC6
Hydrochloric Acid SCHEMBL7016878 0.84 SRC (0.39) TP53MAPTP2RX3RXFP1TSHR
SCHEMBL7019933 0.83 HDAC1 (0.41) TP53MAPTHDAC1HDAC6HDAC2
SCHEMBL7017888 0.83 TP53 (0.47) TP53MAPTP2RX3HDAC1HDAC6
SCHEMBL7010029 0.82 TP53 (0.36) TP53MAPTP2RX3HDAC1HDAC6
SCHEMBL7015809 0.79 HDAC6 (0.48) TP53MAPTHDAC1HDAC6HDAC2
SCHEMBL7015187 0.79 RAB9A (0.37) MAPTP2RX3HDAC1HDAC2TSHR
Hydrochloric Acid SCHEMBL7012711 0.78 PSMB1 (0.49) MAPTTSHRALDH1A1THRBKDM4E
Hydrochloric Acid SCHEMBL7016880 0.77 SMN1; SMN2 (0.46) MAPTHDAC1HDAC6HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed