SCHEMBL7016344

SCHEMBL7016344

O=c1[nH]c2ccc(Cl)cc2c(=O)n1C[C@@H](S)CS

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.56
CA9 Q16790 1/20 0.56
ALDH1A1 P00352 3/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
POLB P06746 2/20 0.53
PKM P14618 1/20 0.53
TBXAS1 P24557 2/20 0.44
CHEK1 O14757 1/20 0.44
AURKA O14965 1/20 0.44
DAPK3 O43293 1/20 0.44
JAK2 O60674 1/20 0.44
MAP4K4 O95819 1/20 0.44
ABL1 P00519 1/20 0.44
NTRK1 P04629 1/20 0.44
LCK P06239 1/20 0.44
CSF1R P07333 1/20 0.44
RET P07949 1/20 0.44
MET P08581 1/20 0.44
PDGFRB P09619 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7019787 0.90 CA9 (0.56) CA12CA9KMT2APKMTBXAS1
SCHEMBL7022854 0.81 CYP1A2 (0.59) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL8987779 0.81 CA12 (0.57) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL8987863 0.78 MPO (0.57) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL11008112 0.76 CA12 (0.59) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL7023017 0.75 KDM4E (0.56) ALDH1A1MEN1KMT2APOLBMPO
SCHEMBL11009308 0.75 CA12 (0.61) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL9049869 0.74 CA12 (0.60) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL14560540 0.73 MPO (0.57) CA12CA9ALDH1A1MEN1KMT2A
SCHEMBL7019436 0.71 TSHR (0.35) ALDH1A1MEN1KMT2APOLBPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003089416-A1 SUBSTITUTED PYRIMIDINE-2,4(1H,3H)-DIONES FOR USE AS MATRIX METALLOPROTEINASE (MMP) INHIBITORS IBFB GMBH (DE) 2003-10-30 WO claimed
EP-1357114-A1 Substituted pyrimidin-2,4(1H,3H)-diones as inhibitors of Matrix Metalloproteinases (MMP) IBFB GmbH Privates Institut für biomedizinische Forschung und Beratung (DE) 2003-10-29 EP claimed
WO-2003089416-A1 SUBSTITUTED PYRIMIDINE-2,4(1H,3H)-DIONES FOR USE AS MATRIX METALLOPROTEINASE (MMP) INHIBITORS IBFB GMBH (DE) 2003-10-30 WO disclosed
EP-1357114-A1 Substituted pyrimidin-2,4(1H,3H)-diones as inhibitors of Matrix Metalloproteinases (MMP) IBFB GmbH Privates Institut für biomedizinische Forschung und Beratung (DE) 2003-10-29 EP disclosed