SCHEMBL7016752

SCHEMBL7016752

COc1[c]cc(-c2cc3ncncc3[nH]2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.35
CCNB2 O95067 4/20 0.35
CDK1 P06493 4/20 0.35
CCNB1 P14635 4/20 0.35
GSK3A P49840 4/20 0.35
GSK3B P49841 4/20 0.35
CCNB3 Q8WWL7 4/20 0.35
CDK5 Q00535 2/20 0.35
CDK5R1 Q15078 2/20 0.35
FGFR4 P22455 1/20 0.34
KDM4E B2RXH2 2/20 0.33
NR3C1 P04150 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
FGFR3 P22607 2/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
CASP3 P42574 1/20 0.31
RAB9A P51151 1/20 0.31
SENP8 Q96LD8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7019380 0.80 RIPK1 (0.41) EGFRCCNB2CDK1CCNB1GSK3A
SCHEMBL7103387 0.76 KDM4E (0.39) CCNB2CDK1CCNB1CCNB3CDK5
SCHEMBL7019407 0.75 CCNB2 (0.38) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL6286092 0.74 ALDH1A1 (0.41) FGFR4KDM4ENR3C1ALDH1A1HPGD
SCHEMBL14976218 0.71 CCNB2 (0.49) EGFRCCNB2CDK1CCNB1GSK3A
SCHEMBL6286089 0.70 ACVR1 (0.42) KDM4ENR3C1ALDH1A1HPGD
SCHEMBL6494995 0.69 KDM4E (0.38) CCNB2CDK1CCNB1CCNB3KDM4E
SCHEMBL6287089 0.67 SMN1; SMN2 (0.51) KDM4EALDH1A1HPGD
SCHEMBL6287083 0.65 NPY5R (0.41) EGFRKDM4ENR3C1ALDH1A1HPGD
SCHEMBL7019826 0.65 RIPK1 (0.42) CCNB2CDK1CCNB1GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294718-A2 6,5-FUSED BICYCLIC HETEROCYCLES WARNER-LAMBERT COMPANY LLC (US) 2003-03-26 EP claimed
WO-2001096336-A2 6,5-FUSED BICYCLIC HETEROCYCLES WARNER-LAMBERT COMPANY (US) 2001-12-20 WO claimed