SCHEMBL7103387

SCHEMBL7103387

COc1[c]cc(-c2cc3cnncc3[nH]2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
MAPT P10636 2/20 0.39
CASP3 P42574 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
CCNA2 P20248 5/20 0.36
CDK2 P24941 5/20 0.36
TTK P33981 5/20 0.36
AURKA O14965 4/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
FYN P06241 2/20 0.35
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
CCNB2 O95067 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6494995 0.79 KDM4E (0.38) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL7019407 0.77 CCNB2 (0.38) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL7019826 0.77 RIPK1 (0.42) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL7019380 0.76 RIPK1 (0.41) CCNA2CDK2TTKAURKACCNB2
SCHEMBL7016752 0.76 EGFR (0.35) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL6286924 0.71 CYP1A1 (0.44) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL7104266 0.68 PDGFRB (0.38) KDM4EMAPTMEN1KMT2AALDH1A1
SCHEMBL6286918 0.67 PARP1 (0.47) CCNA2CDK2TTKAURKAFYN
SCHEMBL7100815 0.64 RIPK1 (0.42) KDM4ENPC1RAB9AMAPTCASP3
SCHEMBL4820299 0.62 ESR2 (0.48) KDM4ENPC1RAB9AMAPTCASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294718-A2 6,5-FUSED BICYCLIC HETEROCYCLES WARNER-LAMBERT COMPANY LLC (US) 2003-03-26 EP disclosed
WO-2001096336-A2 6,5-FUSED BICYCLIC HETEROCYCLES WARNER-LAMBERT COMPANY (US) 2001-12-20 WO disclosed