SCHEMBL7017547

SCHEMBL7017547

CCOC(=O)c1ccccc1C(=O)c1ccc(CBr)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.62
CYP4F2 P78329 1/20 0.54
CYP4A11 Q02928 1/20 0.54
CDC25B P30305 1/20 0.54
ALDH1A1 P00352 8/20 0.51
L3MBTL1 Q9Y468 4/20 0.51
NPSR1 Q6W5P4 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
HSD17B10 Q99714 2/20 0.50
LMNA P02545 4/20 0.49
THRB P10828 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
HPGD P15428 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29121130 0.89 TSHR (0.68) TSHRCDC25BALDH1A1L3MBTL1NPSR1
SCHEMBL420 0.85 CES2 (0.49) TSHRALDH1A1L3MBTL1NPSR1CYP1A2
SCHEMBL4463486 0.84 TSHR (0.70) TSHRCDC25BALDH1A1L3MBTL1NPSR1
SCHEMBL29619268 0.84 TSHR (0.75) TSHRCDC25BALDH1A1L3MBTL1NPSR1
SCHEMBL195278 0.84 TSHR (0.75) TSHRCDC25BALDH1A1L3MBTL1NPSR1
SCHEMBL9541280 0.84 CES2 (0.62) TSHRCDC25BALDH1A1L3MBTL1NPSR1
SCHEMBL4733061 0.83 TSHR (0.68) TSHRCDC25BALDH1A1L3MBTL1NPSR1
SCHEMBL9356956 0.82 TSHR (0.66) TSHRCDC25BALDH1A1L3MBTL1NPSR1
SCHEMBL10429982 0.81 ALDH1A1 (0.45) ALDH1A1L3MBTL1NPSR1CYP1A2CYP3A4
SCHEMBL245250 0.81 CA1 (0.63) TSHRCYP4F2CYP4A11ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed