SCHEMBL9541280

SCHEMBL9541280

O=C(c1ccc(CBr)cc1)c1ccccc1C(=O)c1ccc(CBr)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.62
CES1 P23141 1/20 0.62
AKR1C3 P42330 3/20 0.53
CDC25B P30305 2/20 0.50
ATM Q13315 1/20 0.50
NR4A1 P22736 1/20 0.48
LIG1 P18858 1/20 0.47
ALDH1A1 P00352 4/20 0.46
TSHR P16473 2/20 0.46
TRPA1 O75762 1/20 0.46
CDC25A P30304 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7011648 0.87 KMT2A (0.57) CES2CES1AKR1C3NR4A1ALDH1A1
SCHEMBL420 0.87 CES2 (0.49) CES2CES1ATMALDH1A1TSHR
SCHEMBL118227 0.85 CES2 (0.77) CES2CES1ATMALDH1A1TSHR
SCHEMBL187134 0.84 CES2 (0.61) CES2CES1ALDH1A1TSHRTRPA1
SCHEMBL9541276 0.84 CES2 (0.61) CES2CES1ALDH1A1TSHRTRPA1
SCHEMBL7017547 0.84 TSHR (0.62) CES2CES1CDC25BALDH1A1TSHR
SCHEMBL7017613 0.83 STS (0.56) CES2CES1ATMALDH1A1HSD17B10
SCHEMBL10429982 0.83 ALDH1A1 (0.45) CES2CES1AKR1C3ALDH1A1CYP1A2
Dimethylamine SCHEMBL6131311 0.82 CES2 (0.67) CES2CES1ATMALDH1A1TSHR
SCHEMBL1041339 0.81 CES2 (0.54) CES2CES1AKR1C3CDC25BATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993005028-A1 RECEPTOR COMPOUNDS BASED ON 1,7-DIOXA-4,10-DIAZACYCLODODECANE SCIMAT LIMITED (GB) 1993-03-18 WO disclosed