SCHEMBL7017613

SCHEMBL7017613

COc1ccccc1C(=O)c1ccc(CBr)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STS P08842 1/20 0.56
ATM Q13315 1/20 0.52
RAB9A P51151 4/20 0.51
NPC1 O15118 3/20 0.51
MAPT P10636 3/20 0.50
ALDH1A1 P00352 1/20 0.50
CTSD P07339 1/20 0.49
CES2 O00748 1/20 0.49
CES1 P23141 1/20 0.49
HPGD P15428 2/20 0.48
KMT2A Q03164 1/20 0.48
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
RXRA P19793 1/20 0.47
TP53 P04637 1/20 0.47
GLA P06280 1/20 0.47
GAA P10253 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KDM4E B2RXH2 1/20 0.45
ALOX15 P16050 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9541280 0.83 CES2 (0.62) ATMMAPTALDH1A1CES2CES1
SCHEMBL26988530 0.82 KMT2A (0.68) STSRAB9ANPC1MAPTALDH1A1
SCHEMBL6616664 0.82 MAPT (0.69) STSATMRAB9ANPC1MAPT
SCHEMBL3484026 0.82 RAB9A (0.66) STSRAB9ANPC1MAPTALDH1A1
SCHEMBL50229 0.81 MAPT (0.64) STSATMRAB9ANPC1MAPT
SCHEMBL29573531 0.81 MAPT (0.64) STSATMRAB9ANPC1MAPT
SCHEMBL420 0.81 CES2 (0.49) ATMMAPTALDH1A1CES2CES1
SCHEMBL1584218 0.80 RAB9A (0.67) STSRAB9ANPC1MAPTALDH1A1
SCHEMBL1682193 0.80 STS (0.70) STSRAB9ANPC1MAPTALDH1A1
SCHEMBL31286496 0.80 RAB9A (0.67) STSRAB9ANPC1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed