SCHEMBL7017972

SCHEMBL7017972

N#Cc1c(N)nc(OCc2cccnc2)c(C#N)c1-c1c(F)cccc1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
HSD17B10 Q99714 4/20 0.49
MAPK1 P28482 3/20 0.49
SQOR Q9Y6N5 1/20 0.48
ADORA1 P30542 7/20 0.44
KDM4E B2RXH2 7/20 0.43
GAA P10253 2/20 0.43
HPGD P15428 2/20 0.43
MGMT P16455 1/20 0.43
GLA P06280 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ADORA2A P29274 3/20 0.42
ADORA3 P0DMS8 1/20 0.42
HTT P42858 2/20 0.41
TSHR P16473 2/20 0.41
RXFP1 Q9HBX9 1/20 0.40
ROCK2 O75116 1/20 0.40
CSF1R P07333 1/20 0.40
MAPK8 P45983 1/20 0.40
MAPK9 P45984 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7018457 0.89 ALDH1A1 (0.64) ALDH1A1HSD17B10MAPK1SQORADORA1
SCHEMBL3545741 0.84 RXFP1 (0.55) ALDH1A1HSD17B10MAPK1SQORADORA1
SCHEMBL7019882 0.78 SQOR (0.45) HSD17B10MAPK1SQORADORA1KDM4E
SCHEMBL26010519 0.77 ADORA1 (0.52) ALDH1A1HSD17B10MAPK1SQORADORA1
SCHEMBL7024723 0.77 ALDH1A1 (0.67) ALDH1A1HSD17B10MAPK1SQORADORA1
SCHEMBL3554945 0.76 ADORA2A (0.52) ALDH1A1HSD17B10MAPK1SQORADORA1
SCHEMBL1154965 0.75 HTR1A (0.49) ALDH1A1SQORKDM4EHPGDSMN1; SMN2
SCHEMBL7022211 0.75 GSK3A (0.55) ALDH1A1HSD17B10MAPK1SQORADORA1
SCHEMBL3550981 0.71 ADORA1 (0.60) ALDH1A1HSD17B10MAPK1SQORADORA1
SCHEMBL6442682 0.71 HSD17B10 (0.62) ALDH1A1HSD17B10MAPK1SQORADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1302463-A1 MEDICINE COMPRISING DICYANOPYRIDINE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 2003-04-16 EP disclosed