SCHEMBL7018034

SCHEMBL7018034

O=C(c1ccc(Cl)cc1)c1ccc(Cn2ccn3c(=O)c4c(nc23)CCC4)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.42
HSD17B10 Q99714 3/20 0.42
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 2/20 0.42
PIK3CD O00329 1/20 0.42
PIK3CB P42338 1/20 0.42
PKM P14618 1/20 0.42
TP53 P04637 5/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
LMNA P02545 4/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
MMP13 P45452 1/20 0.40
KMT2A Q03164 5/20 0.39
MAPT P10636 5/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016280 0.99 PIK3CD (0.43) HPGDHSD17B10ALDH1A1KDM4EPIK3CD
SCHEMBL7015344 0.89 PIK3CD (0.43) HPGDHSD17B10ALDH1A1KDM4EPIK3CD
SCHEMBL7017560 0.85 ALDH1A1 (0.36) HPGDHSD17B10ALDH1A1KDM4EPIK3CD
SCHEMBL7015959 0.78 TP53 (0.44) ALDH1A1PIK3CDPIK3CBTP53HDAC3
SCHEMBL7015350 0.76 TP53 (0.44) PIK3CDPIK3CBTP53HDAC3HDAC1
SCHEMBL7016621 0.76 TP53 (0.42) ALDH1A1PIK3CDPIK3CBPKMTP53
SCHEMBL7014282 0.75 TP53 (0.41) PIK3CDPIK3CBTP53HDAC3HDAC1
SCHEMBL7016868 0.74 ENPP2 (0.42) HSD17B10ALDH1A1KDM4EPIK3CDPIK3CB
SCHEMBL7016044 0.74 PIK3CD (0.55) KDM4EPIK3CDPIK3CBTP53HDAC3
SCHEMBL7018099 0.73 LMNA (0.50) HPGDALDH1A1KDM4ETP53LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed