SCHEMBL7018995

SCHEMBL7018995

Cc1nc2[nH]ccn2c(=O)c1C

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM5B Q9UGL1 1/20 0.35
BRD4 O60885 2/20 0.34
RAB9A P51151 5/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KDM4E B2RXH2 2/20 0.33
NPC1 O15118 4/20 0.33
ALDH1A1 P00352 2/20 0.31
HPGD P15428 1/20 0.31
CYP1A2 P05177 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
TAF1 P21675 1/20 0.30
BRPF1 P55201 1/20 0.30
CREBBP Q92793 1/20 0.30
CECR2 Q9BXF3 1/20 0.30
BRD9 Q9H8M2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27311213 0.82 TDP1 (0.49) KDM5BBRD4RAB9ASMN1; SMN2NPC1
SCHEMBL24097994 0.82 BRD4 (0.33) BRD4
SCHEMBL7017850 0.80 KDM5B (0.59) KDM5BRAB9ASMN1; SMN2KDM4ENPC1
SCHEMBL7016511 0.80 KDM5B (0.44) KDM5BBRD4SMN1; SMN2
SCHEMBL31661272 0.73 KMT2A (0.50) RAB9ASMN1; SMN2KDM4EALDH1A1CYP1A2
SCHEMBL19779493 0.70 ADORA3 (0.39) KDM5BRAB9ASMN1; SMN2KDM4ENPC1
SCHEMBL23335815 0.70 KDM4E (0.46) KDM5BBRD4SMN1; SMN2KDM4EALDH1A1
SCHEMBL31661243 0.68 SMN1; SMN2 (0.35) BRD4SMN1; SMN2KDM4EALDH1A1HPGD
SCHEMBL24236934 0.68 BRD9 (0.39) BRD4KDM4EALDH1A1CYP1A2TAF1
SCHEMBL7015921 0.67 KDM4E (0.54) RAB9ASMN1; SMN2KDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed