SCHEMBL7019229

SCHEMBL7019229

CN(C)Cc1nc2[c]cccc2[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.38
TDP1 Q9NUW8 1/20 0.37
CYP3A4 P08684 2/20 0.36
MAPT P10636 1/20 0.36
PIM1 P11309 3/20 0.35
PIM2 Q9P1W9 3/20 0.35
DDAH1 O94760 1/20 0.34
MAPK14 Q16539 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MYC P01106 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
HSD17B10 Q99714 2/20 0.33
TSHR P16473 2/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
ACHE P22303 1/20 0.31
ADRB2 P07550 1/20 0.31
PIM3 Q86V86 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7021216 0.81 DDAH1 (0.53) MAPTDDAH1ALDH1A1HSD17B10TSHR
SCHEMBL7024978 0.79 DDAH1 (0.39) MAPTDDAH1KMT2AKDM4EPOLB
SCHEMBL7019566 0.78 TDP1 (0.40) BCHETDP1DDAH1MEN1KMT2A
SCHEMBL7017120 0.78 CACNA1H (0.36) BCHEDDAH1PKMPOLB
SCHEMBL908058 0.78 DDAH1 (0.33) BCHEDDAH1ALDH1A1HSD17B10KDM4E
SCHEMBL7017479 0.77 NPC1 (0.39) MAPTDDAH1ALDH1A1MEN1KMT2A
SCHEMBL7014749 0.75 LMNA (0.33) BCHECYP3A4MAPTALDH1A1MEN1
SCHEMBL698519 0.74 GAA (0.58) TDP1MAPTKMT2ATSHRKDM4E
SCHEMBL9598374 0.74 MEN1 (0.33) MAPTDDAH1ALDH1A1MEN1KMT2A
SCHEMBL11719783 0.74 POLB (0.45) ALDH1A1PKMPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051415-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 2003-09-24 EP disclosed
US-6495542-B1 SUCH AS 2-METHOXY-N-(2-METHYL-1H-BENZIMIDAZOL-4-YL)-4-(2,3,4,5-TETRAHYDRO-5-OXO-1H-1-BENZAZEPIN-1-YL)CARBONYL-BENZAM IDE; HYPERTENSION, HEART FAILURE, RENAL INSUFFICIENCY, EDEMA, ASCITES, VASOPRESSIN PARASECRETION SYNDROME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-12-17 US disclosed