SCHEMBL7019995

SCHEMBL7019995

COc1cc(N)c(C(=O)O)cc1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.53
ALDH1A1 P00352 3/20 0.51
LCK P06239 1/20 0.46
FYN P06241 1/20 0.46
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.43
KMT2A Q03164 3/20 0.43
TDP1 Q9NUW8 3/20 0.43
MEN1 O00255 2/20 0.43
IDO1 P14902 1/20 0.43
MYC P01106 1/20 0.42
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41
CA14 Q9ULX7 2/20 0.41
GFER P55789 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
HTT P42858 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29918238 1.00 KDM4E (0.53) KDM4EALDH1A1LCKFYNGAA
SCHEMBL3125277 0.93 KDM4E (0.53) KDM4EALDH1A1LCKFYNGAA
SCHEMBL22691985 0.87 ALDH1A1 (0.58) KDM4EALDH1A1LCKFYNGAA
SCHEMBL85946 0.86 KDM4E (0.69) KDM4EALDH1A1LCKFYNGAA
SCHEMBL10520470 0.85 KDM4E (0.53) KDM4EALDH1A1GAACA9HTT
SCHEMBL3549850 0.85 KDM4E (0.53) KDM4EALDH1A1GAAHPGDHTT
Hydrochloric Acid SCHEMBL5012089 0.85 KDM4E (0.67) KDM4EALDH1A1LCKFYNGAA
SCHEMBL23520824 0.84 KDM4E (0.77) KDM4EALDH1A1GAAHPGDHTT
Nitrogen SCHEMBL28644623 0.83 KDM4E (0.65) KDM4EALDH1A1LCKFYNGAA
SCHEMBL13596372 0.82 ALDH1A1 (0.56) KDM4EALDH1A1LCKFYNHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102850397-B Multi-target antitumor compounds and preparation method and application thereof UNIV BEIJING 2015-02-18 CN claimed
CN-102850397-A Multi-target antitumor compounds and preparation method and application thereof UNIV BEIJING 2013-01-02 CN claimed
CN-102850397-B Multi-target antitumor compounds and preparation method and application thereof UNIV BEIJING 2015-02-18 CN disclosed
CN-102850397-A Multi-target antitumor compounds and preparation method and application thereof UNIV BEIJING 2013-01-02 CN disclosed
WO-2003106435-A1 FUSED-RING PYRIMIDIN-4(3H)-ONE DERIVATIVES, PROCESSES FOR THE PREPARATION AND USES THEREOF SANKYO COMPANY, LIMITED (JP) 2003-12-24 WO disclosed