SCHEMBL7024075

SCHEMBL7024075

CC(C)(C)OC(=O)Nc1cc(-c2[c]cccc2C(F)(F)F)ccn1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 10/20 0.42
CYP3A4 P08684 4/20 0.42
IRAK4 Q9NWZ3 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
TGFBR1 P36897 1/20 0.40
PIK3C3 Q8NEB9 2/20 0.39
NR3C2 P08235 1/20 0.39
TRPV1 Q8NER1 1/20 0.37
GSK3B P49841 1/20 0.37
DYRK1A Q13627 1/20 0.37
IGF1R P08069 1/20 0.37
PHGDH O43175 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6992479 0.87 IRAK4 (0.42) AAK1CYP3A4IRAK4TGFBR1PIK3C3
SCHEMBL5225197 0.86 TGFBR1 (0.43) AAK1CYP3A4IRAK4TGFBR1PIK3C3
SCHEMBL7026837 0.85 IRAK4 (0.42) AAK1IRAK4TGFBR1PIK3C3GSK3B
SCHEMBL6990608 0.84 AAK1 (0.41) AAK1IRAK4TGFBR1PIK3C3NR3C2
SCHEMBL7020508 0.80 TGFBR1 (0.40) AAK1CYP3A4IRAK4TGFBR1PIK3C3
SCHEMBL5251219 0.75 EGFR (0.57) AAK1IRAK4TGFBR1PIK3C3GSK3B
SCHEMBL5812808 0.75 RIPK3 (0.41) AAK1IRAK4TGFBR1PIK3C3GSK3B
SCHEMBL29992322 0.72 AAK1 (0.48) AAK1CYP3A4IRAK4TGFBR1PIK3C3
SCHEMBL8670718 0.72 FDPS (0.50) AAK1CYP3A4IRAK4TGFBR1PIK3C3
SCHEMBL17643492 0.72 AAK1 (0.48) AAK1CYP3A4IRAK4TGFBR1PIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268474-A2 SUBSTITUTED 1,3-THIAZOLE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2003-01-02 EP disclosed
WO-2001074811-A2 SUBSTITUTED 1,3-THIAZOLE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-10-11 WO disclosed