SCHEMBL7026883

SCHEMBL7026883

CN(C(=O)C(CC1CCCCC1)NC(=O)c1cccc(Oc2ccccc2)c1)C1(C#N)CCNCC1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 11/20 0.52
CTSL P07711 10/20 0.52
CTSK P43235 4/20 0.48
CTSB P07858 4/20 0.48
GPR132 Q9UNW8 1/20 0.44
PKM P14618 1/20 0.42
NPY5R Q15761 1/20 0.41
ALDH1A1 P00352 2/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPC1 O15118 1/20 0.39
MEN1 O00255 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
RAB9A P51151 1/20 0.38
CHRM3 P20309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7417185 0.91 CTSL (0.57) CTSSCTSLCTSKCTSB
SCHEMBL7422431 0.86 CTSS (0.47) CTSSCTSLCTSKCTSBGPR132
SCHEMBL7410718 0.82 CTSS (0.47) CTSSCTSLCTSKCTSBNPC1
SCHEMBL7409657 0.82 CTSS (0.60) CTSSCTSLCTSKCTSBGPR132
SCHEMBL7414009 0.81 USP30 (0.46) CTSSCTSLCTSKCTSBALDH1A1
SCHEMBL7414894 0.80 CTSS (0.45) CTSSCTSLCTSKCTSB
SCHEMBL7414674 0.79 CTSS (0.45) CTSSCTSLCTSKCTSBALDH1A1
SCHEMBL5528965 0.78 CTSL (0.79) CTSSCTSLCTSKCTSBGPR132
SCHEMBL5365066 0.75 CTSS (0.57) CTSSCTSLCTSKCTSBGPR132
SCHEMBL7423676 0.75 CTSL (0.44) CTSSCTSLCTSKCTSBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003529546-A 2003-10-07 JP claimed
EP-1218372-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-07-03 EP claimed
WO-2001019816-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-03-22 WO claimed