SCHEMBL7417185

SCHEMBL7417185

CN(C(=O)C(CC1CCCCC1)NC(=O)c1ccccc1)C1(C#N)CCNCC1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSL P07711 12/20 0.57
CTSS P25774 11/20 0.57
CTSB P07858 5/20 0.57
CTSK P43235 3/20 0.57
CHRNB2 P17787 2/20 0.43
CHRNB4 P30926 2/20 0.43
CHRNA3 P32297 2/20 0.43
CHRNA4 P43681 2/20 0.43
USP30 Q70CQ3 2/20 0.43
CTSV O60911 2/20 0.41
GRN P28799 1/20 0.40
SORT1 Q99523 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRM1 Q13255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7410718 0.91 CTSS (0.47) CTSLCTSSCTSBCTSKCHRNB2
SCHEMBL7409657 0.91 CTSS (0.60) CTSLCTSSCTSBCTSKCHRNB2
SCHEMBL7026883 0.91 CTSS (0.52) CTSLCTSSCTSBCTSK
SCHEMBL7414894 0.89 CTSS (0.45) CTSLCTSSCTSBCTSKUSP30
SCHEMBL7414009 0.88 USP30 (0.46) CTSLCTSSCTSBCTSKCHRNB2
SCHEMBL7414674 0.87 CTSS (0.45) CTSLCTSSCTSBCTSKUSP30
SCHEMBL7423676 0.83 CTSL (0.44) CTSLCTSSCTSBCTSK
SCHEMBL7414874 0.80 CTSS (0.46) CTSLCTSSCTSBCTSKCHRNB2
SCHEMBL5525335 0.80 CTSL (0.69) CTSLCTSSCTSBCTSKCHRNB2
SCHEMBL5530441 0.80 CTSL (0.69) CTSLCTSSCTSBCTSKCHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218372-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-07-03 EP disclosed
WO-2001019816-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-03-22 WO disclosed