SCHEMBL7027236

SCHEMBL7027236

COc1cc[c]c(-c2ccnc(NC(=O)OC(C)(C)C)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3C3 Q8NEB9 2/20 0.42
AAK1 Q2M2I8 11/20 0.40
IRAK4 Q9NWZ3 1/20 0.40
ATR Q13535 1/20 0.39
TGFBR1 P36897 1/20 0.39
RIOK2 Q9BVS4 1/20 0.39
NR3C2 P08235 1/20 0.39
ROCK2 O75116 2/20 0.38
NR2C2 P49116 2/20 0.38
HIPK4 Q8NE63 2/20 0.38
BMP2K Q9NSY1 2/20 0.38
GAK O14976 1/20 0.38
CHRNA1 P02708 1/20 0.38
SLC6A2 P23975 1/20 0.38
CHRNA7 P36544 1/20 0.38
TAB1 Q15750 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
GSK3B P49841 1/20 0.38
DYRK1A Q13627 1/20 0.38
MAP2K1 Q02750 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5812808 0.88 RIPK3 (0.41) PIK3C3AAK1IRAK4ATRTGFBR1
SCHEMBL7026492 0.84 TGFBR1 (0.41) PIK3C3AAK1IRAK4ATRTGFBR1
SCHEMBL3938343 0.82 RIOK2 (0.51) ATRRIOK2NR3C2HIPK4MKNK2
SCHEMBL30427105 0.82 RIOK2 (0.51) ATRRIOK2NR3C2HIPK4MKNK2
SCHEMBL12127932 0.81 FDPS (0.54) PIK3C3AAK1RIOK2NR3C2GSK3B
SCHEMBL7492460 0.80 MAPK14 (0.54) RIOK2
SCHEMBL7020508 0.77 TGFBR1 (0.40) PIK3C3AAK1IRAK4ATRTGFBR1
SCHEMBL5251219 0.74 EGFR (0.57) PIK3C3AAK1IRAK4TGFBR1RIOK2
SCHEMBL5225197 0.74 TGFBR1 (0.43) PIK3C3AAK1IRAK4ATRTGFBR1
SCHEMBL17155229 0.74 AAK1 (0.49) PIK3C3AAK1IRAK4ATRROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268474-A2 SUBSTITUTED 1,3-THIAZOLE COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2003-01-02 EP disclosed
WO-2001074811-A2 SUBSTITUTED 1,3-THIAZOLE COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-10-11 WO disclosed