SCHEMBL7028358

SCHEMBL7028358

CC(C)(C)C(=O)Oc1ccc2[nH]c(=O)[nH]c(=O)c2c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 1/20 0.48
HTR1B P28222 1/20 0.48
ELANE P08246 12/20 0.46
PDE3B Q13370 1/20 0.44
PDE3A Q14432 1/20 0.44
GABRA1 P14867 1/20 0.43
GABRG2 P18507 1/20 0.43
GABRB3 P28472 1/20 0.43
CA12 O43570 2/20 0.42
CA9 Q16790 2/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PARP1 P09874 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7024662 0.84 PDE3B (0.53) HTR1DPDE3BPDE3ACA12CA9
SCHEMBL7027645 0.80 HTR1A (0.50) HTR1DHTR1BELANEPDE3BPDE3A
SCHEMBL7029183 0.79 KIF11 (0.50) PDE3BPDE3ACA12CA9KDM4E
SCHEMBL3792832 0.79 PARP15 (0.54) PDE3BPDE3ACA12CA9KDM4E
SCHEMBL3124589 0.77 ALDH1A1 (0.63) CA12CA9KDM4EALDH1A1HPGD
SCHEMBL7023220 0.76 LIMK1 (0.55) CA12CA9KDM4EALDH1A1MEN1
SCHEMBL7029348 0.76 PDE3B (0.48) HTR1BPDE3BPDE3AKDM4EALDH1A1
SCHEMBL8821061 0.74 GABRA1 (0.48) HTR1DHTR1BELANEGABRA1GABRG2
SCHEMBL7031912 0.73 CA12 (0.46) PDE3BPDE3ACA12CA9KDM4E
SCHEMBL7030752 0.73 KDM4E (0.60) PDE3BPDE3ACA12CA9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0878468-B1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL CO (JP) 2003-03-19 EP disclosed
EP-0775697-B1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL CO (JP) 2003-02-12 EP disclosed
US-5994542-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-11-30 US disclosed
EP-0878468-A1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-11-18 EP disclosed
US-5756738-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-05-26 US disclosed
EP-0775697-A1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-05-28 EP disclosed