SCHEMBL7031087

SCHEMBL7031087

O=C(c1ccccc1)c1c(Cl)cc2c3c1c1c(n3CCC2=O)CCNCC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.35
HTR2A P28223 5/20 0.35
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
RORC P51449 1/20 0.33
SIGMAR1 Q99720 1/20 0.32
KDM4E B2RXH2 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
HPGD P15428 1/20 0.31
CASP1 P29466 1/20 0.31
CYP2C19 P33261 1/20 0.31
HTR6 P50406 2/20 0.31
HTR2B P41595 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
PARP1 P09874 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7036280 0.88 HTR2C (0.35) HTR2CHTR2AUSP2ALDH1A1TSHR
SCHEMBL7038309 0.82 HTR6 (0.38) HTR2CHTR2AUSP2ALDH1A1TSHR
Oxalic Acid SCHEMBL6496558 0.73 HTR2C (0.44) HTR2CHTR2AALDH1A1KDM4EHTR6
Oxalic Acid SCHEMBL6492860 0.71 HTR2C (0.52) HTR2CHTR2AHSD17B10SIGMAR1KDM4E
SCHEMBL6507807 0.70 HTR2C (0.48) HTR2CHTR2AHSD17B10KDM4EHTR6
SCHEMBL6507779 0.69 HTR2C (0.58) HTR2CHTR2AHSD17B10SIGMAR1KDM4E
SCHEMBL7033472 0.69 RORC (0.31) HTR2CHTR2AUSP2ALDH1A1TSHR
SCHEMBL7033915 0.68 HTR2C (0.34) HTR2CHTR2AUSP2ALDH1A1TSHR
SCHEMBL6498327 0.67 PTGDR2 (0.45) USP2ALDH1A1HPGDMEN1KMT2A
Fumaric Acid SCHEMBL6499043 0.65 HTR2C (0.37) HTR2CHTR2AALDH1A1HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173440-B1 TETRACYCLIC AZEPINOINDOLE COMPOUNDS AS 5-HT RECEPTOR LIGANDS UPJOHN CO (US) 2004-09-15 EP claimed