SCHEMBL7036280

SCHEMBL7036280

O=C(c1ccccc1)c1c(F)cc2c3c1c1c(n3CCC2=O)CCNCC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.35
HTR2A P28223 4/20 0.35
TSHR P16473 2/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HSD17B10 Q99714 1/20 0.34
RORC P51449 1/20 0.33
HPGD P15428 3/20 0.33
NPC1 O15118 1/20 0.33
TP53 P04637 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPK1 P28482 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
SIGMAR1 Q99720 1/20 0.32
KDM4E B2RXH2 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CASP1 P29466 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7031087 0.88 HTR2C (0.35) HTR2CHTR2ATSHRUSP2ALDH1A1
SCHEMBL7038309 0.82 HTR6 (0.38) HTR2CHTR2ATSHRUSP2ALDH1A1
SCHEMBL7033472 0.81 RORC (0.31) HTR2CHTR2ATSHRUSP2ALDH1A1
Oxalic Acid SCHEMBL6492860 0.71 HTR2C (0.52) HTR2CHTR2AHSD17B10TP53ALOX15
SCHEMBL6498458 0.69 HTR2C (0.40) HTR2CHTR2AHSD17B10ALOX15MAPK1
Maleic Acid SCHEMBL6495798 0.69 HTR2C (0.35) HTR2CHTR2ASIGMAR1HTR6
Fumaric Acid SCHEMBL6495804 0.69 HTR2C (0.35) HTR2CHTR2ASIGMAR1HTR6
SCHEMBL6507779 0.69 HTR2C (0.58) HTR2CHTR2AHSD17B10TP53ALOX15
Oxalic Acid SCHEMBL6496558 0.68 HTR2C (0.44) HTR2CHTR2AALDH1A1KDM4EHTR6
SCHEMBL6507807 0.66 HTR2C (0.48) HTR2CHTR2AHSD17B10ALOX15MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173440-B1 TETRACYCLIC AZEPINOINDOLE COMPOUNDS AS 5-HT RECEPTOR LIGANDS UPJOHN CO (US) 2004-09-15 EP claimed