SCHEMBL7032072

SCHEMBL7032072

CC(C)(C)OC(=O)N1CCC(CCCC(=O)Nc2nnn[nH]2)CC1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.52
GPR119 Q8TDV5 14/20 0.51
GLS O94925 2/20 0.48
KDM4E B2RXH2 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3477072 0.74 FAAH (0.56) FAAHGPR119KDM4EPKM
SCHEMBL15085741 0.74 GPR119 (0.59) FAAHGPR119KDM4EPKM
SCHEMBL3476578 0.73 FAAH (0.55) FAAHGPR119GLS
SCHEMBL6794692 0.73 FAAH (0.56) FAAHGPR119KDM4EPKM
SCHEMBL20077080 0.73 FAAH (0.58) FAAHGPR119KDM4EPKM
SCHEMBL13999420 0.73 FAAH (0.58) FAAHGPR119KDM4EPKM
SCHEMBL544238 0.73 FAAH (0.58) FAAHGPR119KDM4EPKM
SCHEMBL2539468 0.72 GPR119 (0.67) FAAHGPR119
SCHEMBL3478015 0.72 FAAH (0.57) FAAHGPR119KDM4EPKM
SCHEMBL459905 0.71 MAPT (0.51) GPR119KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040092737-A1 Benzopiperidine derivatives EISAI CO., LTD. 2004-05-13 US disclosed
US-6518423-B1 These compounds are useful as drugs efficacious in the prevention and treatment of these various inflammatory diseases and immunologic diseases, such as rheumatoid arthritis, atopic dermatitis, psoriasis, asthma, and EISAI CO., LTD. (JP) 2003-02-11 US disclosed
EP-0934941-A1 BENZOPIPERIDINE DERIVATIVES Eisai Co., Ltd. (JP) 1999-08-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040092737-A1 Benzopiperidine derivatives HLA-DRB1, HRH1, HRH2 FAAH 604/4885GPR119 1119/4885GLS 2045/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.