SCHEMBL7033172

SCHEMBL7033172

O=C(c1ccccc1)c1ccc2c3c1c1c(n3C(C(F)(F)F)CC2=O)CCNCC1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.35
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
PARP1 P09874 1/20 0.31
USP2 O75604 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CYP2C8 P10632 1/20 0.30
CYP2C9 P11712 1/20 0.30
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7037088 0.83 HTR6 (0.34) HTR6HTR2CPARP1
Oxalic Acid SCHEMBL6496999 0.80 HTR6 (0.38) HTR6HTR2AHTR2CHSD17B10
SCHEMBL7038309 0.78 HTR6 (0.38) HTR6HTR2AHTR2CPARP1USP2
SCHEMBL7033472 0.72 RORC (0.31) HTR2AHTR2CUSP2ALDH1A1TSHR
SCHEMBL7038313 0.68 HTR2C (0.38) HTR6HTR2AHTR2CPARP1HSD17B10
SCHEMBL7033915 0.66 HTR2C (0.34) HTR6HTR2AHTR2CUSP2ALDH1A1
SCHEMBL7036278 0.65 HTR6 (0.35) HTR6HTR2AHTR2CHSD17B10
Oxalic Acid SCHEMBL6496099 0.64 HTR2C (0.42) HTR6HTR2AHTR2CALDH1A1HSD17B10
SCHEMBL7033168 0.64 HTR6 (0.35) HTR6HTR2AHTR2CPARP1HSD17B10
SCHEMBL7031084 0.63 HTR6 (0.35) HTR6HTR2AHTR2CHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173440-B1 TETRACYCLIC AZEPINOINDOLE COMPOUNDS AS 5-HT RECEPTOR LIGANDS UPJOHN CO (US) 2004-09-15 EP claimed