SCHEMBL7038510

SCHEMBL7038510

CCc1cc(OC(N)=O)c2nc(N3CCNCC3)[nH]c2c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.37
HRH4 Q9H3N8 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
PARP1 P09874 11/20 0.37
HTR3A P46098 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
HTR6 P50406 1/20 0.35
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
DRD3 P35462 1/20 0.35
TP53 P04637 1/20 0.35
NAMPT P43490 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7045004 0.96 PIM1 (0.38) KCNH2HRH4HRH3PARP1HTR3A
SCHEMBL7037681 0.84 HTR3A (0.39) PARP1HTR3ANAMPT
SCHEMBL7043691 0.83 HTR3A (0.39) PARP1HTR3ATP53NAMPT
SCHEMBL5622568 0.83 PARP1 (0.50) PARP1
SCHEMBL7045539 0.81 CHRNB2 (0.40) HRH4PARP1HTR3A
SCHEMBL7042860 0.80 PIM1 (0.41) HRH4PARP1HTR3ANAMPT
SCHEMBL5620205 0.80 PARP1 (0.47) PARP1
SCHEMBL7039844 0.80 CHRNB2 (0.42) HRH4PARP1HTR3ATP53NAMPT
SCHEMBL7041756 0.80 CHRNB2 (0.43) HRH4PARP1HTR3A
SCHEMBL6869623 0.78 PARP1 (0.49) PARP1HTR3AHTR6NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed