SCHEMBL7042860

SCHEMBL7042860

NC(=O)Oc1cc(N)cc2[nH]c(N3CCCNCC3)nc12

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 2/20 0.41
CHRNB2 P17787 2/20 0.39
CHRNA4 P43681 2/20 0.39
PARP1 P09874 10/20 0.36
HTR3A P46098 1/20 0.36
HRH4 Q9H3N8 1/20 0.36
CHRNA1 P02708 1/20 0.35
CHRNA7 P36544 1/20 0.35
ENPP1 P22413 1/20 0.35
NAMPT P43490 1/20 0.34
IKBKB O14920 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7037681 0.96 HTR3A (0.39) PIM1PARP1HTR3ANAMPT
SCHEMBL7039844 0.88 CHRNB2 (0.42) PIM1CHRNB2CHRNA4PARP1HTR3A
SCHEMBL7041756 0.88 CHRNB2 (0.43) PIM1CHRNB2CHRNA4PARP1HTR3A
SCHEMBL7045539 0.86 CHRNB2 (0.40) PIM1CHRNB2CHRNA4PARP1HTR3A
SCHEMBL7045004 0.85 PIM1 (0.38) PIM1CHRNB2CHRNA4PARP1HTR3A
SCHEMBL6864445 0.83 PARP1 (0.46) PIM1PARP1HTR3A
SCHEMBL7043691 0.83 HTR3A (0.39) PIM1CHRNB2CHRNA4PARP1HTR3A
SCHEMBL5620167 0.83 PARP1 (0.50) CHRNB2CHRNA4PARP1
SCHEMBL7038510 0.80 KCNH2 (0.37) PARP1HTR3AHRH4NAMPT
SCHEMBL6869623 0.78 PARP1 (0.49) PARP1HTR3ANAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed