SCHEMBL7045004

SCHEMBL7045004

CCc1cc(OC(N)=O)c2nc(N3CCCNCC3)[nH]c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.38
CHRNB2 P17787 2/20 0.36
CHRNA4 P43681 2/20 0.36
ENPP1 P22413 1/20 0.36
IKBKB O14920 1/20 0.36
PARP1 P09874 7/20 0.35
KCNH2 Q12809 1/20 0.35
HRH4 Q9H3N8 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
HTR3A P46098 1/20 0.34
PRKD1 Q15139 1/20 0.34
PRKD2 Q9BZL6 1/20 0.34
TP53 P04637 1/20 0.33
HTR6 P50406 1/20 0.33
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
HTR2A P28223 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7038510 0.96 KCNH2 (0.37) PARP1KCNH2HRH4HRH3ITGB3
SCHEMBL7042860 0.85 PIM1 (0.41) PIM1CHRNB2CHRNA4ENPP1IKBKB
SCHEMBL7039844 0.85 CHRNB2 (0.42) PIM1CHRNB2CHRNA4ENPP1PARP1
SCHEMBL5620205 0.85 PARP1 (0.47) PARP1
SCHEMBL7041756 0.85 CHRNB2 (0.43) PIM1CHRNB2CHRNA4PARP1HRH4
SCHEMBL7045539 0.82 CHRNB2 (0.40) PIM1CHRNB2CHRNA4PARP1HRH4
SCHEMBL7037681 0.81 HTR3A (0.39) PIM1PARP1HTR3A
SCHEMBL6864445 0.80 PARP1 (0.46) PIM1PARP1HTR3A
SCHEMBL7043691 0.80 HTR3A (0.39) PIM1CHRNB2CHRNA4PARP1HTR3A
SCHEMBL5622568 0.80 PARP1 (0.50) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed