SCHEMBL7039533

SCHEMBL7039533

O=C(O)c1cccc2ncc(-c3ccc(Br)cc3)nc12

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.60
PARP2 Q9UGN5 1/20 0.56
ALDH1A1 P00352 1/20 0.49
RXFP1 Q9HBX9 1/20 0.47
EPRS1 P07814 4/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1034874 0.88 PARP1 (0.62) PARP1PARP2ALDH1A1
SCHEMBL7042977 0.88 PARP1 (0.78) PARP1PARP2RXFP1
SCHEMBL7044628 0.84 PARP1 (0.60) PARP1PARP2ALDH1A1
SCHEMBL31353202 0.77 PARP1 (0.59) PARP1PARP2ALDH1A1
SCHEMBL7111338 0.77 PARP1 (0.80) PARP1PARP2ALDH1A1
SCHEMBL7039537 0.76 AURKA (0.51) PARP1ALDH1A1
SCHEMBL1033372 0.76 PARP1 (0.62) PARP1PARP2ALDH1A1
SCHEMBL7112515 0.75 PARP1 (1.00) PARP1PARP2
SCHEMBL7113559 0.75 PARP1 (0.67) PARP1PARP2ALDH1A1RXFP1
SCHEMBL24186148 0.74 ALDH1A1 (0.59) PARP1PARP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003007959-A1 QUINOXALINE DERIVATIVES WHICH HAVE PARP INHIBITORY ACTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-30 WO disclosed