SCHEMBL7112515

SCHEMBL7112515

NC(=O)c1cccc2ncc(-c3ccc(N)cc3)nc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 1.00
PARP2 Q9UGN5 2/20 0.74
DHODH Q02127 2/20 0.43
TLR9 Q9NR96 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
PKN1 Q16512 1/20 0.41
PKN2 Q16513 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7111338 0.89 PARP1 (0.80) PARP1PARP2DHODHPKN1PKN2
SCHEMBL7045309 0.88 PARP1 (0.78) PARP1PARP2DHODH
SCHEMBL31602072 0.88 PARP1 (0.81) PARP1PARP2DHODHNPC1RAB9A
SCHEMBL424209 0.88 PARP1 (0.81) PARP1PARP2DHODHNPC1RAB9A
SCHEMBL7042977 0.88 PARP1 (0.78) PARP1PARP2DHODH
SCHEMBL7108289 0.85 PARP1 (1.00) PARP1PARP2
SCHEMBL7045177 0.84 PARP1 (1.00) PARP1PARP2NPC1RAB9A
SCHEMBL7107333 0.84 PARP1 (1.00) PARP1PARP2
SCHEMBL7043497 0.83 PARP1 (0.71) PARP1PARP2DHODHPKN1PKN2
SCHEMBL7042013 0.83 PARP1 (0.71) PARP1PARP2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003007959-A1 QUINOXALINE DERIVATIVES WHICH HAVE PARP INHIBITORY ACTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-30 WO disclosed