SCHEMBL7042977

SCHEMBL7042977

NC(=O)c1cccc2ncc(-c3ccc(Br)cc3)nc12

nearest known ligand 0.78

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.78
PARP2 Q9UGN5 2/20 0.73
RXFP1 Q9HBX9 2/20 0.44
CASP1 P29466 1/20 0.44
KMT2A Q03164 1/20 0.43
CSF1R P07333 1/20 0.42
DHODH Q02127 1/20 0.42
GRM2 Q14416 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7039533 0.88 PARP1 (0.60) PARP1PARP2RXFP1
SCHEMBL7112515 0.88 PARP1 (1.00) PARP1PARP2DHODH
SCHEMBL7111338 0.87 PARP1 (0.80) PARP1PARP2DHODH
SCHEMBL7113559 0.87 PARP1 (0.67) PARP1PARP2RXFP1KMT2A
SCHEMBL7045309 0.86 PARP1 (0.78) PARP1PARP2CSF1RDHODHGRM2
SCHEMBL31602072 0.86 PARP1 (0.81) PARP1PARP2CASP1KMT2ADHODH
SCHEMBL424209 0.86 PARP1 (0.81) PARP1PARP2CASP1KMT2ADHODH
SCHEMBL7108289 0.84 PARP1 (1.00) PARP1PARP2CASP1CSF1R
SCHEMBL7044628 0.83 PARP1 (0.60) PARP1PARP2KMT2A
SCHEMBL7107333 0.83 PARP1 (1.00) PARP1PARP2CASP1CSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003007959-A1 QUINOXALINE DERIVATIVES WHICH HAVE PARP INHIBITORY ACTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-30 WO disclosed