SCHEMBL7040201

SCHEMBL7040201

CN1CCC(c2nc3c(OC(N)=O)cccc3n2C)CC1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.54
HTR2B P41595 1/20 0.43
PARP2 Q9UGN5 2/20 0.39
HSD11B1 P28845 1/20 0.36
TLR7 Q9NYK1 1/20 0.35
ITGB3 P05106 3/20 0.35
ITGAV P06756 3/20 0.35
HTR1A P08908 1/20 0.35
HTR1B P28222 1/20 0.35
HTR1F P30939 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
PDE10A Q9Y233 1/20 0.34
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7040671 0.93 PARP1 (0.50) PARP1HTR2BPARP2HSD11B1CHRM1
SCHEMBL7045615 0.89 PARP1 (0.51) PARP1HTR2BPARP2
SCHEMBL7042003 0.87 PARP1 (0.48) PARP1HTR2BPARP2TLR7MEN1
SCHEMBL7038340 0.86 PARP1 (0.48) PARP1HTR2BHSD11B1MEN1KMT2A
SCHEMBL7043510 0.85 PARP1 (0.55) PARP1HTR2BMEN1KMT2A
SCHEMBL7043780 0.85 PARP1 (0.47) PARP1HTR2BPARP2HSD11B1
SCHEMBL7040495 0.85 PARP1 (0.65) PARP1PARP2
SCHEMBL7043077 0.83 PARP1 (0.44) PARP1HTR2BPARP2CHRM1
SCHEMBL7044945 0.83 PARP1 (0.45) PARP1HTR2BHSD11B1
SCHEMBL7041082 0.82 PARP1 (0.52) PARP1HTR2BMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed