SCHEMBL7044945

SCHEMBL7044945

CC(=O)N1CCCC(c2nc3c(OC(N)=O)cccc3n2C)C1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.45
PROKR1 Q8TCW9 2/20 0.42
HSD11B1 P28845 1/20 0.39
BTK Q06187 2/20 0.38
ADORA2A P29274 3/20 0.37
HTR2B P41595 1/20 0.37
HTR2A P28223 1/20 0.36
TMEM97 Q5BJF2 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
PDE4B Q07343 1/20 0.35
PDE7A Q13946 1/20 0.35
CHEK2 O96017 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7038340 0.95 PARP1 (0.48) PARP1PROKR1HSD11B1BTKHTR2B
SCHEMBL7040671 0.85 PARP1 (0.50) PARP1PROKR1HSD11B1HTR2B
SCHEMBL5622558 0.84 PARP1 (0.62) PARP1PROKR1
SCHEMBL7040201 0.83 PARP1 (0.54) PARP1HSD11B1HTR2B
SCHEMBL7043274 0.82 TP53 (0.46) PARP1HSD11B1BTK
SCHEMBL7040495 0.82 PARP1 (0.65) PARP1
SCHEMBL7043780 0.82 PARP1 (0.47) PARP1HSD11B1HTR2B
SCHEMBL7042003 0.80 PARP1 (0.48) PARP1HTR2B
SCHEMBL7041082 0.79 PARP1 (0.52) PARP1HTR2BALDH1A1
SCHEMBL7044651 0.79 MEN1 (0.40) PDE7AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed