SCHEMBL7042964

SCHEMBL7042964

NC(=O)Oc1cccc2c1nc(N1CCNCC1)n2CCO

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 7/20 0.42
SOS1 Q07889 1/20 0.37
HTR2C P28335 2/20 0.37
PIM1 P11309 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7044695 0.96 HTR3A (0.40) HTR3ASOS1HTR2CPIM1
SCHEMBL7042935 0.92 HTR3A (0.42) HTR3ASOS1HTR2CPIM1KCNH2
SCHEMBL7041296 0.89 HTR3A (0.40) HTR3ASOS1HTR2C
SCHEMBL7041533 0.89 HTR3A (0.40) HTR3A
SCHEMBL7045272 0.88 FLT3 (0.44) HTR3ASOS1PIM1KCNH2
SCHEMBL7036855 0.88 HTR3A (0.40) HTR3ASOS1HTR2CPIM1
SCHEMBL7039363 0.88 HTR3A (0.40) HTR3ASOS1HTR2CKCNH2
SCHEMBL7046613 0.88 HTR3A (0.40) HTR3A
SCHEMBL7046777 0.86 HTR3A (0.39) HTR3A
SCHEMBL7043722 0.85 MEN1 (0.37) HTR3ASOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed