SCHEMBL7045264

SCHEMBL7045264

CSc1ccc(CC=O)cc1F

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 4/20 0.33
LMNA P02545 1/20 0.32
STK17B O94768 1/20 0.32
CCR2 P41597 1/20 0.31
AR P10275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17295058 0.79 TAS1R3 (0.37) SLC6A4
SCHEMBL8372279 0.79 TRPA1 (0.39) SLC6A4LMNA
SCHEMBL2712117 0.78 L3MBTL1 (0.33) SLC6A4LMNA
SCHEMBL17295109 0.77 IDO1 (0.35) CCR2AR
SCHEMBL31451660 0.77 SLC6A4 (0.35) SLC6A4LMNASTK17BAR
SCHEMBL31038741 0.77 LOXL2 (0.41) SLC6A4
SCHEMBL6513914 0.77 SLC6A4 (0.35) SLC6A4LMNASTK17BAR
SCHEMBL6520589 0.77 CYP4F2 (0.42) SLC6A4LMNASTK17BAR
SCHEMBL896163 0.76 HTT (0.42)
SCHEMBL22826739 0.76 CNR1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3148972-A1 PYRAZOLONE DERIVATIVES AS NITROXYL DONORS Cardioxyl Pharmaceuticals Inc. (US) 2017-04-05 EP disclosed
WO-2015183839-A1 PYRAZOLONE DERIVATIVES AS NITROXYL DONORS CARDIOXYL PHARMACEUTICALS, INC. (US) 2015-12-03 WO disclosed
EP-1296971-A2 2-FLUOROBENZENESULFONYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION Pharmacia Corporation (US) 2003-04-02 EP disclosed
WO-2001081332-A2 2-FLUOROBENZENESULFONYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA CORPORATION (US) 2001-11-01 WO disclosed