SCHEMBL7046162

SCHEMBL7046162

CN(C)CC(=O)Nc1nc2cc(OS(=O)(=O)c3ccc(NC4CCCC4)cc3)ccc2[nH]1.O=C(Nc1nc2cc(OS(=O)(=O)c3ccc(-n4ccnc4)cc3)ccc2[nH]1)NC1CC1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SLC6A9 P48067 1/20 0.35
NOS2 P35228 1/20 0.35
CD38 P28907 7/20 0.35
ROCK2 O75116 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
LIPG Q9Y5X9 1/20 0.34
MMP1 P03956 3/20 0.34
PDPK1 O15530 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5040906 0.89 NPC1 (0.46) NPC1RAB9ANOS2CD38MAPT
SCHEMBL5036523 0.88 NPC1 (0.48) NPC1RAB9ANOS2CD38MAPT
SCHEMBL5037996 0.87 NPC1 (0.44) NPC1RAB9ANOS2CD38MAPT
SCHEMBL5043085 0.87 NPC1 (0.41) NPC1RAB9ACD38LIPGMMP1
SCHEMBL5036222 0.87 LMNA (0.38) NOS2CD38MAPTHTTMMP1
SCHEMBL5043014 0.87 ENPP3 (0.39) NPC1RAB9AMAPTHTT
SCHEMBL7050284 0.86 MET (0.36) CD38ROCK2MAPTHTTMMP1
SCHEMBL7176912 0.86 MAPT (0.39) NPC1RAB9AROCK2MAPTHTT
SCHEMBL7049236 0.86 MMP1 (0.38) NPC1RAB9ANOS2ROCK2MAPT
SCHEMBL5033770 0.85 CD38 (0.41) NPC1RAB9ACD38LIPGMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1432417-A2 SUBSTITUTED BENZIMIDAZOLE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF CANCER Aventis Pharma S.A. (FR) 2004-06-30 EP disclosed
WO-2003028721-A2 SUBSTITUTED BENZIMIDAZOLE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF CANCER AVENTIS PHARMA S.A. (FR) 2003-04-10 WO disclosed