SCHEMBL7048665

SCHEMBL7048665

CC(C)(C)OC(=O)NCC(=O)N1CCC[C@]1(C(=O)NCc1ccc(C#N)cc1Cl)C1CCCCC1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 6/20 0.41
ALDH1A1 P00352 2/20 0.40
EPHX2 P34913 6/20 0.38
DRD2 P14416 1/20 0.34
AAK1 Q2M2I8 1/20 0.33
EGLN1 Q9GZT9 1/20 0.33
ENPP2 Q13822 1/20 0.32
JAK3 P52333 1/20 0.32
BTK Q06187 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7049344 0.90 JAK2 (0.39) ALDH1A1EPHX2DRD2AAK1ENPP2
SCHEMBL7045257 0.84 DPP4 (0.37) AAK1JAK3BTK
SCHEMBL7045772 0.81 JAK2 (0.40) ALDH1A1EPHX2ENPP2JAK3
SCHEMBL7045869 0.80 NAMPT (0.40) EGLN1JAK3BTK
SCHEMBL8781179 0.76 DPP4 (0.37) AAK1
SCHEMBL7046882 0.75 JAK2 (0.39) ALDH1A1EPHX2DRD2AAK1ENPP2
SCHEMBL5900915 0.75 MEN1 (0.44) ALDH1A1DRD2BTK
SCHEMBL13780330 0.75 P2RX7 (0.53) P2RX7ALDH1A1EPHX2
SCHEMBL5900918 0.72 MEN1 (0.45) ALDH1A1DRD2BTK
SCHEMBL7048588 0.71 NAMPT (0.39) EGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773955-B1 NEW THROMBIN INHIBITORS, THEIR PREPARATION AND USE BASF AG (DE) 2003-04-16 EP disclosed
EP-0773955-A1 NEW THROMBIN INHIBITORS, THEIR PREPARATION AND USE BASF AKTIENGESELLSCHAFT (DE) 1997-05-21 EP disclosed
WO-1995035309-A1 NEW THROMBIN INHIBITORS, THEIR PREPARATION AND USE BASF AKTIENGESELLSCHAFT (DE) 1995-12-28 WO disclosed