SCHEMBL7046882

SCHEMBL7046882

COc1cc(C#N)ccc1CNC(=O)OC1(C2CCCCC2)CCN1C(=O)CNC(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
JAK3 P52333 1/20 0.39
KDM4D Q6B0I6 1/20 0.38
DRD2 P14416 3/20 0.34
PDE4A P27815 2/20 0.34
PDE4B Q07343 2/20 0.34
PDE4C Q08493 2/20 0.34
PDE4D Q08499 2/20 0.34
ENPP2 Q13822 1/20 0.34
MMP13 P45452 2/20 0.33
MMP2 P08253 1/20 0.33
AAK1 Q2M2I8 1/20 0.33
EPHX2 P34913 1/20 0.33
ALDH1A1 P00352 2/20 0.32
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
FPR3 P25089 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7049344 0.85 JAK2 (0.39) JAK2JAK1TYK2JAK3KDM4D
SCHEMBL23775495 0.77 ABCB1 (0.43) JAK2JAK1TYK2JAK3KDM4D
SCHEMBL30305200 0.77 ABCB1 (0.43) JAK2JAK1TYK2JAK3KDM4D
SCHEMBL7045772 0.77 JAK2 (0.40) JAK2JAK1TYK2JAK3KDM4D
SCHEMBL7048665 0.75 P2RX7 (0.41) JAK3DRD2ENPP2AAK1EPHX2
SCHEMBL7050773 0.71 ALDH1A1 (0.42) JAK2JAK1TYK2JAK3KDM4D
SCHEMBL7047070 0.70 ALDH1A1 (0.64) JAK2JAK1TYK2JAK3EPHX2
SCHEMBL7045257 0.68 DPP4 (0.37) JAK2JAK1JAK3KDM4DAAK1
SCHEMBL5900918 0.68 MEN1 (0.45) DRD2MMP13ALDH1A1MMP1MMP9
SCHEMBL24838783 0.68 TRPV1 (0.44) DRD2ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773955-B1 NEW THROMBIN INHIBITORS, THEIR PREPARATION AND USE BASF AG (DE) 2003-04-16 EP disclosed