SCHEMBL7050853

SCHEMBL7050853

O=[C]c1cccc(C#CCO)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
MELK Q14680 1/20 0.41
MMP2 P08253 1/20 0.39
MMP12 P39900 1/20 0.39
FFAR1 O14842 3/20 0.37
MAPK14 Q16539 1/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
EGFR P00533 1/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP2D6 P10635 1/20 0.36
ALOX5 P09917 1/20 0.34
ASIC3 Q9UHC3 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
THPO P40225 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5633251 0.89 ALDH1A1 (0.47) ALDH1A1MELKMMP2MMP12FFAR1
SCHEMBL32144372 0.80 FFAR1 (0.47) ALDH1A1MELKFFAR1
SCHEMBL82303 0.80 FFAR1 (0.47) ALDH1A1MELKFFAR1
SCHEMBL1070719 0.78 MAPT (0.35) ALDH1A1FFAR1CYP3A4
SCHEMBL25201198 0.78 HSD17B13 (0.47) ALDH1A1MELKFFAR1KDM4ELMNA
SCHEMBL30422943 0.78 HSD17B13 (0.47) ALDH1A1MELKFFAR1KDM4ELMNA
SCHEMBL28886 0.78 APP (0.35) ALDH1A1CYP3A4
SCHEMBL1244860 0.76 FFAR1 (0.51) ALDH1A1MELKMMP2MMP12FFAR1
SCHEMBL79516 0.76 ALDH1A1 (0.41) ALDH1A1MELKMMP2MMP12MAPK14
SCHEMBL79281 0.76 GRM5 (0.50) ALDH1A1MELKFFAR1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102739-B1 GLUCOCORTICOID AND THYROID HORMONE RECEPTOR LIGANDS FOR THE TREATMENT OF METABOLIC DISORDERS KAROBIO AB (SE) 2003-04-23 EP disclosed
US-6492424-B1 Glucocorticoid and thyroid hormone receptor ligands for the treatment of metabolic disorders KARO BIO AB (SE) 2002-12-10 US disclosed